Publications – University of Copenhagen

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Chemical Biology & HTS Facility > Publications

Publications

Wilbek T. S., Skovgaard T., Sorrell F. J., Knapp S., Berthelsen J. and Strømgaard K. (2014) “Identification and Characterization of a Small Molecule Inhibitor of Death-Associated Protein Kinase 1”, ChemBioChem, accepted for publication.

Petersen, D. L., Krejsgaard, T., Berthelsen, J., Fredholm, S., Willerslev-Olsen, A., Sibbesen, N. A.,, Bonefeld C M , Andersen M H , Francavilla C , Olsen J V , Hu T , Zhang M , Wasik M A , Geisler C , Woetmann A  and Odum N . (2014). B-lymphoid tyrosine kinase (Blk) is an oncogene and a potential target for therapy with dasatinib in cutaneous T-cell lymphoma (CTCL). Leukemia. Epub available ahead of publication.

Rudolf, A. F., Skovgaard, T., Knapp, S., Jensen, L. J., & Berthelsen, J. (2014). A comparison of protein kinases inhibitor screening methods using both enzymatic activity and binding affinity determination. PLoS ONE, 9(6),

Kotzsch, A., Skovgaard, T., Buus, U., Andersen, S., Devkota, K., & Berthelsen, J. (2014). A substrate-optimized electrophoretic mobility shift assay for ADAM12. Analytical Biochemistry, 452, 34–42.

Devkota, K., Lohse, B., Liu, Q., Wang, M.-W., Stærk, D., Berthelsen, J., & Clausen, R. P. (2014). Analogues of the Natural Product Sinefungin as Inhibitors of EHMT1 and EHMT2. ACS Medicinal Chemistry Letters, 5(4), 293–297.

Fröhlich C, Klitgaard M, Noer JB, Kotzsch A, Nehammer C, Kronqvist P, Berthelsen J, Blobel C, Kveiborg M, Albrechtsen R, Wewer UM (2013) “ADAM12 is expressed in the tumour vasculature and mediates ectodomain shedding of several membrane-anchored endothelial proteins”. Biochem J. 15; 452(1):97-109.

Lundh M, Christensen DP, Damgaard Nielsen M, Richardson SJ, Dahllöf MS, Skovgaard T, Berthelsen J, Dinarello CA, Stevenazzi A, Mascagni P, Grunnet LG, Morgan NG, Mandrup-Poulsen T. (2012 ) Histone deacetylases 1 and 3 but not 2 mediate cytokine-induced beta cell apoptosis in INS-1 cells and dispersed primary islets from rats and are differentially regulated in the islets of type 1 diabetic children.” Diabetologia. 55(9):2421-31